Applications of Physiologically Based Absorption Models in Drug Discovery and Development

Applications of Physiologically Based Absorption Models in Drug Discovery and Development

Authors: Parrott N, Lavé T
Publication: Mol Pharm
Software: GastroPlus®

This article describes the use of physiologically based models of intestinal drug absorption to guide the research and development of new drugs.

Simulation of Gabapentin Absorption and Bioavailability in Pediatric Patients

Simulation of Gabapentin Absorption and Bioavailability in Pediatric Patients

Conference: ISSX
Division: PBPK

To fit an absorption-pharmacokinetic model for simulation of Gabapentin in adult and pediatric populations. The model will be able to describe the nonlinear dose dependence of absorption mediated by an amino…

Population Pharmacokinetics of Bendamustine and Metabolites in Patients With Indolent Non-Hodgkin Lymphoma

Population Pharmacokinetics of Bendamustine and Metabolites in Patients With Indolent Non-Hodgkin Lymphoma

Conference: ASCPT

Bendamustine is a bifunctional alkylating agent in development as monotherapy and in combination with other agents in the treatment of indolent non-Hodgkin lymphoma (NHL).

Model Feasibility Assessment as a Driver for Model-Based Drug Development

Model Feasibility Assessment as a Driver for Model-Based Drug Development

Conference: ASCPT

Complex pharmacometric analyses raise concerns about cost, time, and reliability of the modelbuilding process (MBP). The goal was to use a model feasibility assessment (MFA) process to improve the performance…

Application of Gastrointestinal Simulation for Extensions for Biowaivers of Highly Permeable Compounds

Application of Gastrointestinal Simulation for Extensions for Biowaivers of Highly Permeable Compounds

Publication: AAPS J
Software: GastroPlus®
Division: PBPK

The goal of this study was to apply gastrointestinal simulation technology and integration of physiological parameters to predict biopharmaceutical drug classification.